Research on new synthetic routes about 114041-16-6

According to the analysis of related databases, 114041-16-6, the application of this compound in the production field has become more and more popular.

Each compound has different characteristics, and only by selecting the characteristics of the compound suitable for a specific situation can the compound be applied on a large scale. 114041-16-6, name is 5,6-Dimethoxyisoindoline, This compound has unique chemical properties. The synthetic route is as follows., COA of Formula: C10H13NO2

A solution of 5,6-dimethoxyisoindoline 10e (0.20 g, 1.13 mmol) in 1,2-dichloroethane (6 mL) is vigorously stirred with 37% aqueous formaldehyde (1.9 mL, 26 mmol) for 5 min. Sodium triacetoxyborohydride (0.72 g, 3.4 mmol) is added in 6 portions over 5 min. The resulting mixture is stirred at room temperature for 3 h. Saturated sodium bicarbonate and dichloromethane are added to the reaction mixture, and the layers are separated. The aqueous layer is extracted with additional dichloromethane (3*). The combined organic phases are washed with water and then brine, dried over Na2SO4 and concentrated under reduced pressure to give crude compound 10f (0.21 g, 100%) as a light-brown solid, m/z=194, [M+H]+

According to the analysis of related databases, 114041-16-6, the application of this compound in the production field has become more and more popular.

Reference:
Patent; Gladius Pharmaceuticals, Inc.; SUTTON, Larry D.; ZAMBONI, Robert; BUREAU, Patrick; HASSANPOUR, Avid; MAMANI LAPARRA, Laura; VIDAL, Marc; WOO, Simon; ZHOU, Nancy; KEENAN, Richard M.; (127 pag.)US2019/100534; (2019); A1;,
Indoline – Wikipedia,
Indoline | C8H9N – PubChem